| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 2A |
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| Ligand | BDBM50171269 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_322148 (CHEMBL883722) |
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| EC50 | 3475±n/a nM |
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| Citation |  Sard, H; Kumaran, G; Morency, C; Roth, BL; Toth, BA; He, P; Shuster, L SAR of psilocybin analogs: discovery of a selective 5-HT 2C agonist. Bioorg Med Chem Lett15:4555-9 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| 5-hydroxytryptamine receptor 2A |
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| Name: | 5-hydroxytryptamine receptor 2A |
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| Synonyms: | 5-HT-2 | 5-HT-2A | 5-HT2A | 5-hydroxytryptamine receptor 2A (5-HT-2A) | 5-hydroxytryptamine receptor 2A (5HT-2A) | 5-hydroxytryptamine receptor 2A (5HT2A) | 5HT2A_HUMAN | HTR2 | HTR2A | Serotonin receptor 2A |
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| Type: | undefined |
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| Mol. Mass.: | 52607.65 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P28223 |
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| Residue: | 471 |
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| Sequence: | MDILCEENTSLSSTTNSLMQLNDDTRLYSNDFNSGEANTSDAFNWTVDSENRTNLSCEGC
LSPSCLSLLHLQEKNWSALLTAVVIILTIAGNILVIMAVSLEKKLQNATNYFLMSLAIAD
MLLGFLVMPVSMLTILYGYRWPLPSKLCAVWIYLDVLFSTASIMHLCAISLDRYVAIQNP
IHHSRFNSRTKAFLKIIAVWTISVGISMPIPVFGLQDDSKVFKEGSCLLADDNFVLIGSF
VSFFIPLTIMVITYFLTIKSLQKEATLCVSDLGTRAKLASFSFLPQSSLSSEKLFQRSIH
REPGSYTGRRTMQSISNEQKACKVLGIVFFLFVVMWCPFFITNIMAVICKESCNEDVIGA
LLNVFVWIGYLSSAVNPLVYTLFNKTYRSAFSRYIQCQYKENKKPLQLILVNTIPALAYK
SSQLQMGQKKNSKQDAKTTDNDCSMVALGKQHSEEASKDNSDGVNEKVSCV
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| BDBM50171269 |
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| n/a |
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| Name | BDBM50171269 |
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| Synonyms: | 3-[2-(dimethylamino)ethyl]-1H-indol-4-yl dihydrogen phosphate | 4-phosphoryloxy-N,N-dimethyltryptamine | CHEMBL194378 | Indocybin | O-phosphoryl-4-hydroxy-N,N-dimethyltryptamine | Psilocybine | US11597738, Example 4 | psilocin phosphate ester | psilocybin |
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| Type | Small organic molecule |
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| Emp. Form. | C12H17N2O4P |
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| Mol. Mass. | 284.2481 |
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| SMILES | CN(C)CCc1c[nH]c2cccc(OP(O)(O)=O)c12 |
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| Structure | 
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