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TargetCoiled-coil domain-containing protein 6
LigandBDBM50601766
Substrate/Competitorn/a
Meas. Tech.ChEMBL_2238126 (CHEMBL5152022)
IC50 0.400000±n/a nM
Citation Saha, DRyan, KRLakkaniga, NRAcharya, BGarcia, NGSmith, ELFrett, B Targeting Rearranged during Transfection in Cancer: A Perspective on Small-Molecule Inhibitors and Their Clinical Development. J Med Chem64:11747-11773 (2021) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Coiled-coil domain-containing protein 6
Name:Coiled-coil domain-containing protein 6
Synonyms:CCDC6 | CCDC6_HUMAN | Coiled-coil domain-containing protein 6 | D10S170 | Papillary thyroid carcinoma-encoded protein | Protein H4 | TST1
Type:PROTEIN
Mol. Mass.:53294.85
Organism:Homo sapiens (Human)
Description:ChEMBL_109661
Residue:474
Sequence:
MADSASESDTDGAGGNSSSSAAMQSSCSSTSGGGGGGGGGGGGGKSGGIVISPFRLEELT
NRLASLQQENKVLKIELETYKLKCKALQEENRDLRKASVTIQARAEQEEEFISNTLFKKI
QALQKEKETLAVNYEKEEEFLTNELSRKLMQLQHEKAELEQHLEQEQEFQVNKLMKKIKK
LENDTISKQLTLEQLRREKIDLENTLEQEQEALVNRLWKRMDKLEAEKRILQEKLDQPVS
APPSPRDISMEIDSPENMMRHIRFLKNEVERLKKQLRAAQLQHSEKMAQYLEEERHMREE
NLRLQRKLQREMERREALCRQLSESESSLEMDDERYFNEMSAQGLRPRTVSSPIPYTPSP
SSSRPISPGLSYASHTVGFTPPTSLTRAGMSYYNSPGLHVQHMGTSHGITRPSPRRSNSP
DKFKRPTPPPSPNTQTPVQPPPPPPPPPMQPTVPSAATSQPTPSQHSAHPSSQP
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50601766
n/a
NameBDBM50601766
Synonyms:CHEMBL5171764
TypeSmall organic molecule
Emp. Form.C27H32FN9O2
Mol. Mass.533.6005
SMILESn/a
Structure
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