| Reaction Details |
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 | Report a problem with these data |
| Target | UDP-glucuronosyltransferase 2B17 |
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| Ligand | BDBM50183602 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_339080 (CHEMBL867716) |
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| IC50 | 305000±n/a nM |
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| Citation |  Bichlmaier, I; Siiskonen, A; Finel, M; Yli-Kauhaluoma, J Stereochemical sensitivity of the human UDP-glucuronosyltransferases 2B7 and 2B17. J Med Chem49:1818-27 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| UDP-glucuronosyltransferase 2B17 |
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| Name: | UDP-glucuronosyltransferase 2B17 |
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| Synonyms: | UDB17_HUMAN | UGT2B17 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 61109.88 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_436440 |
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| Residue: | 530 |
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| Sequence: | MSLKWMSVFLLMQLSCYFSSGSCGKVLVWPTEYSHWINMKTILEELVQRGHEVIVLTSSA
SILVNASKSSAIKLEVYPTSLTKNDLEDFFMKMFDRWTYSISKNTFWSYFSQLQELCWEY
SDYNIKLCEDAVLNKKLMRKLQESKFDVLLADAVNPCGELLAELLNIPFLYSLRFSVGYT
VEKNGGGFLFPPSYVPVVMSELSDQMIFMERIKNMIYMLYFDFWFQAYDLKKWDQFYSEV
LGRPTTLFETMGKAEMWLIRTYWDFEFPRPFLPNVDFVGGLHCKPAKPLPKEMEEFVQSS
GENGIVVFSLGSMISNMSEESANMIASALAQIPQKVLWRFDGKKPNTLGSNTRLYKWLPQ
NDLLGHPKTKAFITHGGTNGIYEAIYHGIPMVGIPLFADQHDNIAHMKAKGAALSVDIRT
MSSRDLLNALKSVINDPIYKENIMKLSRIHHDQPVKPLDRAVFWIEFVMRHKGAKHLRVA
AHNLTWIQYHSLDVIAFLLACVATMIFMITKCCLFCFRKLAKTGKKKKRD
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| BDBM50183602 |
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| n/a |
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| Name | BDBM50183602 |
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| Synonyms: | (+)-(S)-7-Nitro-1-tetralol | CHEMBL378390 |
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| Type | Small organic molecule |
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| Emp. Form. | C10H11NO3 |
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| Mol. Mass. | 193.1992 |
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| SMILES | O[C@H]1CCCc2ccc(cc12)[N+]([O-])=O |
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| Structure | 
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