| Reaction Details |
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 | Report a problem with these data |
| Target | 1-acyl-sn-glycerol-3-phosphate acyltransferase beta |
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| Ligand | BDBM50606912 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2261572 (CHEMBL5216583) |
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| IC50 | 15±n/a nM |
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| Citation |  Shahari, MSB; Dolzhenko, AV A closer look at N Eur J Med Chem241:0 (2022) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| 1-acyl-sn-glycerol-3-phosphate acyltransferase beta |
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| Name: | 1-acyl-sn-glycerol-3-phosphate acyltransferase beta |
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| Synonyms: | 1-acylglycerol-3-phosphate O-acyltransferase beta | AGPAT2 | PLCB_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 30924.09 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_321473 |
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| Residue: | 278 |
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| Sequence: | MELWPCLAAALLLLLLLVQLSRAAEFYAKVALYCALCFTVSAVASLVCLLRHGGRTVENM
SIIGWFVRSFKYFYGLRFEVRDPRRLQEARPCVIVSNHQSILDMMGLMEVLPERCVQIAK
RELLFLGPVGLIMYLGGVFFINRQRSSTAMTVMADLGERMVRENLKVWIYPEGTRNDNGD
LLPFKKGAFYLAVQAQVPIVPVVYSSFSSFYNTKKKFFTSGTVTVQVLEAIPTSGLTAAD
VPALVDTCHRAMRTTFLHISKTPQENGATAGSGVQPAQ
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| BDBM50606912 |
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| n/a |
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| Name | BDBM50606912 |
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| Synonyms: | CHEMBL5219496 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H19N5O |
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| Mol. Mass. | 345.3978 |
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| SMILES | CCc1ccc(Nc2nc(N)nc(n2)-c2oc3ccccc3c2C)cc1 |
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| Structure | 
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