| Reaction Details |
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 | Report a problem with these data |
| Target | D(2) dopamine receptor |
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| Ligand | BDBM50197199 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_408171 (CHEMBL907725) |
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| Ki | 5000±n/a nM |
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| Citation |  Colabufo, NA; Berardi, F; Perrone, R; Rapposelli, S; Digiacomo, M; Balsamo, A Arylmethyloxyphenyl derivatives: small molecules displaying P-glycoprotein inhibition. J Med Chem49:6607-13 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(2) dopamine receptor |
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| Name: | D(2) dopamine receptor |
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| Synonyms: | D(2) dopamine receptor | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2 | DRD2_HUMAN | Dopamine D2 receptor | Dopamine D2 receptor (D2) | Dopamine D2 receptor (D2R) | Dopamine D2A | Dopamine2-like | d2 |
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| Type: | Cell-surface receptors |
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| Mol. Mass.: | 50647.10 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P14416 |
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| Residue: | 443 |
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| Sequence: | MDPLNLSWYDDDLERQNWSRPFNGSDGKADRPHYNYYATLLTLLIAVIVFGNVLVCMAVS
REKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTA
SILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMISIVWVLSFTISCPLLFGLNNADQN
ECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRRRRKRVNTKRSSRAFRAHLRAPL
KGNCTHPEDMKLCTVIMKSNGSFPVNRRRVEAARRAQELEMEMLSSTSPPERTRYSPIPP
SHHQLTLPDPSHHGLHSTPDSPAKPEKNGHAKDHPKIAKIFEIQTMPNGKTRTSLKTMSR
RKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSA
VNPIIYTTFNIEFRKAFLKILHC
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| BDBM50197199 |
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| n/a |
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| Name | BDBM50197199 |
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| Synonyms: | 1-(benzyloxy)-2-(2-phenylethyl)benzene | 1-(benzyloxy)-2-phenethylbenzene | CHEMBL215010 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H20O |
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| Mol. Mass. | 288.3829 |
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| SMILES | C(Cc1ccccc1OCc1ccccc1)c1ccccc1 |
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| Structure | 
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