| Reaction Details |
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 | Report a problem with these data |
| Target | Apoptosis regulator BAX |
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| Ligand | BDBM50610525 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2281422 |
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| Kd | 255±n/a nM |
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| Citation |  Pogmore, JP; Uehling, D; Andrews, DW Pharmacological Targeting of Executioner Proteins: Controlling Life and Death. J Med Chem64:5276-5290 (2021) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Apoptosis regulator BAX |
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| Name: | Apoptosis regulator BAX |
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| Synonyms: | Apoptosis regulator BAX | BAX | BAX_HUMAN | BCL2L4 | Bcl-2-like protein 4 | Bcl2-L-4 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 21181.15 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_100916 |
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| Residue: | 192 |
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| Sequence: | MDGSGEQPRGGGPTSSEQIMKTGALLLQGFIQDRAGRMGGEAPELALDPVPQDASTKKLS
ECLKRIGDELDSNMELQRMIAAVDTDSPREVFFRVAADMFSDGNFNWGRVVALFYFASKL
VLKALCTKVPELIRTIMGWTLDFLRERLLGWIQDQGGWDGLLSYFGTPTWQTVTIFVAGV
LTASLTIWKKMG
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| BDBM50610525 |
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| n/a |
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| Name | BDBM50610525 |
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| Synonyms: | CHEMBL4578793 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H26N4O |
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| Mol. Mass. | 398.5001 |
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| SMILES | CN1CCN(CC1)C(c1c(-c2ccccc2)n(O)c2ccccc12)c1ccccn1 |
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| Structure | 
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