| Reaction Details |
|---|
 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
|---|
| Ligand | BDBM50220546 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_457315 (CHEMBL941848) |
|---|
| Ki | 13000±n/a nM |
|---|
| Citation |  Stark, D; Piel, M; Hübner, H; Gmeiner, P; Gründer, G; Rösch, F In vitro affinities of various halogenated benzamide derivatives as potential radioligands for non-invasive quantification of D(2)-like dopamine receptors. Bioorg Med Chem15:6819-29 (2007) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| D(1A) dopamine receptor |
|---|
| Name: | D(1A) dopamine receptor |
|---|
| Synonyms: | DRD1 | DRD1_PIG | Dopamine D1 receptor |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 49269.92 |
|---|
| Organism: | Sus scrofa |
|---|
| Description: | ChEMBL_1460140 |
|---|
| Residue: | 446 |
|---|
| Sequence: | MRTLNTSTMDGTGLVVERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTN
FFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVD
RYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNVTSLG
KTTHNCDSSLSRTYAISSSLISFYIPVAIMIVTYTRIYRIAQKQIRRISALERAAVHAKN
CQTTAGNGNPAECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCMVPFCGS
GETKPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPTSTNAIET
VSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIASPLEKLSPAL
SVILDYDTDVSLEKIQPITQNGQHPT
|
|
|
|---|
| BDBM50220546 |
|---|
| n/a |
|---|
| Name | BDBM50220546 |
|---|
| Synonyms: | CHEMBL397103 | N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2-methoxybenzamide |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H21IN2O2 |
|---|
| Mol. Mass. | 400.2546 |
|---|
| SMILES | COc1ccc(I)cc1C(=O)NC[C@@H]1CCCN1CC=C |
|---|
| Structure | 
|
|---|
Search and Browse
