| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 5 |
|---|
| Ligand | BDBM50227101 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_452331 (CHEMBL902568) |
|---|
| Ki | 3950±n/a nM |
|---|
| Citation |  Martin, RE; Green, LG; Guba, W; Kratochwil, N; Christ, A Discovery of the first nonpeptidic, small-molecule, highly selective somatostatin receptor subtype 5 antagonists: a chemogenomics approach. J Med Chem50:6291-4 (2007) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 5 |
|---|
| Name: | Somatostatin receptor type 5 |
|---|
| Synonyms: | SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 39218.02 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P35346 |
|---|
| Residue: | 364 |
|---|
| Sequence: | MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTL
VIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDG
VNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADV
QEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRR
RSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCAN
PVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQ
TSKL
|
|
|
|---|
| BDBM50227101 |
|---|
| n/a |
|---|
| Name | BDBM50227101 |
|---|
| Synonyms: | CHEMBL236787 | N-(1-((1H-indol-5-yl)methyl)piperidin-4-yl)-1-(4-fluorobenzyl)-1H-benzo[d]imidazol-2-amine |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C28H28FN5 |
|---|
| Mol. Mass. | 453.5538 |
|---|
| SMILES | Fc1ccc(Cn2c(NC3CCN(Cc4ccc5[nH]ccc5c4)CC3)nc3ccccc23)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
