| Reaction Details |
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 | Report a problem with these data |
| Target | Phospholipase A2, membrane associated |
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| Ligand | BDBM50262842 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_489271 (CHEMBL990827) |
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| IC50 | 60±n/a nM |
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| Citation |  Oslund, RC; Cermak, N; Gelb, MH Highly specific and broadly potent inhibitors of mammalian secreted phospholipases A2. J Med Chem51:4708-14 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Phospholipase A2, membrane associated |
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| Name: | Phospholipase A2, membrane associated |
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| Synonyms: | PA2GA_MOUSE | Pla2g2a |
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| Type: | PROTEIN |
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| Mol. Mass.: | 16162.44 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_352635 |
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| Residue: | 146 |
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| Sequence: | MKVLLLLAASIMAFGSIQVQGNIAQFGEMIRLKTGKRAELSYAFYGCHCGLGGKGSPKDA
TDRCCVTHDCCYKSLEKSGCGTKLLKYKYSHQGGQITCSANQNSCQKRLCQCDKAAAECF
ARNKKTYSLKYQFYPNMFCKGKKPKC
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| BDBM50262842 |
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| n/a |
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| Name | BDBM50262842 |
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| Synonyms: | Benzenesulfonyl-2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-indol-4-yloxy)acetamide | CHEMBL514692 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H25N3O6S |
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| Mol. Mass. | 519.569 |
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| SMILES | CCc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccccc3)cccc2n1Cc1ccccc1 |
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| Structure | 
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