| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Phospholipase A2 group V |
|---|
| Ligand | BDBM50055391 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_489278 (CHEMBL990834) |
|---|
| IC50 | 44±n/a nM |
|---|
| Citation |  Oslund, RC; Cermak, N; Gelb, MH Highly specific and broadly potent inhibitors of mammalian secreted phospholipases A2. J Med Chem51:4708-14 (2008) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Phospholipase A2 group V |
|---|
| Name: | Phospholipase A2 group V |
|---|
| Synonyms: | PA2G5_HUMAN | PLA2G5 | Phospholipase A2 group V | Secretory phospholipase A2, group V (sPLA2-V) |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 15682.61 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | n/a |
|---|
| Residue: | 138 |
|---|
| Sequence: | MKGLLPLAWFLACSVPAVQGGLLDLKSMIEKVTGKNALTNYGFYGCYCGWGGRGTPKDGT
DWCCWAHDHCYGRLEEKGCNIRTQSYKYRFAWGVVTCEPGPFCHVNLCACDRKLVYCLKR
NLRSYNPQYQYFPNILCS
|
|
|
|---|
| BDBM50055391 |
|---|
| n/a |
|---|
| Name | BDBM50055391 |
|---|
| Synonyms: | 2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-indol-4-yloxy)propanoic acid | 2-(3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-propionic acid | CHEMBL148649 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C22H22N2O5 |
|---|
| Mol. Mass. | 394.4205 |
|---|
| SMILES | CCc1c(C(=O)C(N)=O)c2c(OC(C)C(O)=O)cccc2n1Cc1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
