| Reaction Details |
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 | Report a problem with these data |
| Target | Group 10 secretory phospholipase A2 |
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| Ligand | BDBM50263000 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_489280 (CHEMBL990836) |
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| IC50 | 90±n/a nM |
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| Citation |  Oslund, RC; Cermak, N; Gelb, MH Highly specific and broadly potent inhibitors of mammalian secreted phospholipases A2. J Med Chem51:4708-14 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Group 10 secretory phospholipase A2 |
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| Name: | Group 10 secretory phospholipase A2 |
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| Synonyms: | Group X secretory phospholipase A2 | PA2GX_HUMAN | PLA2G10 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 18153.11 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1442449 |
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| Residue: | 165 |
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| Sequence: | MGPLPVCLPIMLLLLLPSLLLLLLLPGPGSGEASRILRVHRRGILELAGTVGCVGPRTPI
AYMKYGCFCGLGGHGQPRDAIDWCCHGHDCCYTRAEEAGCSPKTERYSWQCVNQSVLCGP
AENKCQELLCKCDQEIANCLAQTEYNLKYLFYPQFLCEPDSPKCD
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| BDBM50263000 |
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| n/a |
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| Name | BDBM50263000 |
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| Synonyms: | 2-(1-benzyl-2-ethyl-1H-6,7-benzoindol-4-yloxy)-N-(phenylsulfonyl)acetamide | CHEMBL446349 |
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| Type | Small organic molecule |
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| Emp. Form. | C31H27N3O6S |
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| Mol. Mass. | 569.628 |
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| SMILES | CCc1c(C(=O)C(N)=O)c2c(OCC(=O)NS(=O)(=O)c3ccccc3)cc3ccccc3c2n1Cc1ccccc1 |
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| Structure | 
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