| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet-activating factor receptor |
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| Ligand | BDBM50284410 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_162886 (CHEMBL768982) |
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| IC50 | 84±n/a nM |
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| Citation |  Chung, SK; Ban, SH; Kim, SH; Kim, BE; Woo, SH; Summers, JB; Conway, RG Synthesis and bioactivities of heterocyclic lipids as PAF antagonists. 2 Bioorg Med Chem Lett5:1097-1102 (1995) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet-activating factor receptor |
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| Name: | Platelet-activating factor receptor |
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| Synonyms: | PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor |
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| Type: | Protein |
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| Mol. Mass.: | 39005.63 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 342 |
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| Sequence: | MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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| BDBM50284410 |
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| n/a |
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| Name | BDBM50284410 |
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| Synonyms: | 1-Ethyl-2-{[(4-methoxy-benzoyl)-(4-octadecylcarbamoyloxymethyl-thietan-2-ylmethoxycarbonyl)-amino]-methyl}-pyridinium; chloride | CHEMBL12556 |
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| Type | Small organic molecule |
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| Emp. Form. | C41H64N3O6S |
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| Mol. Mass. | 727.028 |
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| SMILES | CCCCCCCCCCCCCCCCCCNC(=O)OC[C@H]1C[C@H](COC(=O)N(Cc2cccc[n+]2CC)C(=O)c2ccc(OC)cc2)S1 |
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| Structure | 
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