| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet-activating factor receptor |
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| Ligand | BDBM50284417 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_151708 (CHEMBL760601) |
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| Ki | 5.7±n/a nM |
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| Citation |  Chung, SK; Ban, SH; Kim, SH; Kim, BE; Woo, SH; Summers, JB; Conway, RG Synthesis and bioactivities of heterocyclic lipids as PAF antagonists. 2 Bioorg Med Chem Lett5:1097-1102 (1995) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet-activating factor receptor |
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| Name: | Platelet-activating factor receptor |
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| Synonyms: | PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor |
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| Type: | Protein |
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| Mol. Mass.: | 39005.63 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 342 |
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| Sequence: | MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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| BDBM50284417 |
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| n/a |
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| Name | BDBM50284417 |
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| Synonyms: | 2-{[Acetyl-((2R,4R)-4-octadecylcarbamoyloxymethyl-oxetan-2-ylmethoxycarbonyl)-amino]-methyl}-1-ethyl-pyridinium; iodide | CHEMBL12554 |
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| Type | Small organic molecule |
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| Emp. Form. | C35H60N3O6 |
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| Mol. Mass. | 618.8669 |
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| SMILES | CCCCCCCCCCCCCCCCCCNC(=O)OC[C@H]1C[C@H](COC(=O)N(Cc2cccc[n+]2CC)C(C)=O)O1 |
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| Structure | 
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