| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet-activating factor receptor |
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| Ligand | BDBM50284421 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_151708 (CHEMBL760601) |
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| Ki | 99±n/a nM |
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| Citation |  Chung, SK; Ban, SH; Kim, SH; Kim, BE; Woo, SH; Summers, JB; Conway, RG Synthesis and bioactivities of heterocyclic lipids as PAF antagonists. 2 Bioorg Med Chem Lett5:1097-1102 (1995) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet-activating factor receptor |
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| Name: | Platelet-activating factor receptor |
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| Synonyms: | PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor |
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| Type: | Protein |
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| Mol. Mass.: | 39005.63 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 342 |
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| Sequence: | MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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| BDBM50284421 |
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| n/a |
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| Name | BDBM50284421 |
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| Synonyms: | 1-Ethyl-2-{[((2S,4S)-4-hexadecyloxymethyl-thietan-2-ylmethoxycarbonyl)-(4-methoxy-benzoyl)-amino]-methyl}-pyridinium; chloride | CHEMBL268965 |
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| Type | Small organic molecule |
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| Emp. Form. | C38H59N2O5S |
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| Mol. Mass. | 655.95 |
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| SMILES | CCCCCCCCCCCCCCCCOC[C@@H]1C[C@@H](COC(=O)N(Cc2cccc[n+]2CC)C(=O)c2ccc(OC)cc2)S1 |
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| Structure | 
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