| Reaction Details |
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 | Report a problem with these data |
| Target | D(3) dopamine receptor |
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| Ligand | BDBM50290201 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_58781 |
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| Ki | >7900±n/a nM |
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| Citation |  He, XS; Woodruff, K; Brodbeck, R A new series of selective dopamine D4 ligands: 3-([4-arylpiperazin-1-yl]alkylamino)-2H-1,4-benzoxazines Bioorg Med Chem Lett7:2399-2402 (1997) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(3) dopamine receptor |
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| Name: | D(3) dopamine receptor |
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| Synonyms: | DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3 |
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| Type: | n/a |
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| Mol. Mass.: | 44243.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 400 |
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| Sequence: | MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTV
CSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQ
QTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRK
LSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHV
SPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
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| BDBM50290201 |
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| n/a |
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| Name | BDBM50290201 |
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| Synonyms: | (2H-Benzo[1,4]oxazin-3-yl)-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-butyl]-amine; compound with but-2-enedioic acid | CHEMBL309843 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H26N6O |
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| Mol. Mass. | 366.46 |
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| SMILES | C(CCN1CCN(CC1)c1ncccn1)CNC1=Nc2ccccc2OC1 |t:19| |
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| Structure | 
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