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TargetMetallo-beta-lactamase L1 type 3
LigandBDBM50322613
Substrate/Competitorn/a
Meas. Tech.ChEMBL_641774 (CHEMBL1177097)
Ki 4000±n/a nM
Citation Lassaux, PHamel, MGulea, MDelbrück, HMercuri, PSHorsfall, LDehareng, DKupper, MFrère, JMHoffmann, KGalleni, MBebrone, C Mercaptophosphonate compounds as broad-spectrum inhibitors of the metallo-beta-lactamases. J Med Chem53:4862-76 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Metallo-beta-lactamase L1 type 3
Name:Metallo-beta-lactamase L1 type 3
Synonyms:BLA1_STEMA | Beta-lactamase L1
Type:PROTEIN
Mol. Mass.:30803.13
Organism:Stenotrophomonas maltophilia
Description:ChEMBL_1500319
Residue:290
Sequence:
MRSTLLAFALAVALPAAHTSAAEVPLPQLRAYTVDASWLQPMAPLQIADHTWQIGTEDLT
ALLVQTPDGAVLLDGGMPQMASHLLDNMKARGVTPRDLRLILLSHAHADHAGPVAELKRR
TGAKVAANAESAVLLARGGSDDLHFGDGITYPPANADRIVMDGEVITVGGIVFTAHFMAG
HTPGSTAWTWTDTRNGKPVRIAYADSLSAPGYQLQGNPRYPHLIEDYRRSFATVRALPCD
VLLTPHPGASNWDYAAGARAGAKALTCKAYADAAEQKFDGQLAKETAGAR
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  Blast E-value cutoff:
BDBM50322613
n/a
NameBDBM50322613
Synonyms:CHEMBL1173798 | alpha-Sulfanyl(2-methoxybenzyl)phosphonic acid
TypeSmall organic molecule
Emp. Form.C8H11O4PS
Mol. Mass.234.209
SMILESCOc1ccccc1C(=S)P(O)(O)O
Structure
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