| Reaction Details |
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 | Report a problem with these data |
| Target | Peptide deformylase |
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| Ligand | BDBM50131311 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_154179 |
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| IC50 | 10±n/a nM |
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| Citation |  Davies, SJ; Ayscough, AP; Beckett, RP; Clements, JM; Doel, S; Pratt, LM; Spavold, ZM; Thomas, SW; Whittaker, M Structure--activity relationships of the peptide deformylase inhibitor BB-3497: modification of the P2' and P3' side chains. Bioorg Med Chem Lett13:2715-8 (2003) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Peptide deformylase |
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| Name: | Peptide deformylase |
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| Synonyms: | 3.5.1.88 | BON69_24600 | BON94_18585 | D9G11_24945 | D9G11_25760 | D9J60_20755 | FORC82_p394 | PDF | Polypeptide deformylase | SAMEA3472033_04733 | def | def_2 |
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| Type: | n/a |
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| Mol. Mass.: | 16901.39 |
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| Organism: | Escherichia coli |
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| Description: | n/a |
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| Residue: | 150 |
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| Sequence: | MSVLQVLHIPDERLRKVAKPVEEVNAEIQRIVDDMFETMYAEKGIGLAATQVDIHQRIIV
IDVSENRDERLVLINPELLEKSGETGIEEGCLSIPEQRALVPRAEKVKIRALDRDGKPFE
LEADGLLAICIGLRLGNGKYCTLRLFFNQV
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| BDBM50131311 |
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| n/a |
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| Name | BDBM50131311 |
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| Synonyms: | 1-((S)-2-{(R)-2-[(Formyl-hydroxy-amino)-methyl]-hexanoylamino}-3,3-dimethyl-butyryl)-piperidine-4-carboxylic acid ethyl ester | CHEMBL329677 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H39N3O6 |
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| Mol. Mass. | 441.5616 |
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| SMILES | CCCC[C@H](CN(O)C=O)C(=O)N[C@H](C(=O)N1CCC(CC1)C(=O)OCC)C(C)(C)C |
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| Structure | 
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