| Reaction Details |
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 | Report a problem with these data |
| Target | Sigma non-opioid intracellular receptor 1 |
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| Ligand | BDBM50017039 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_201888 |
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| IC50 | 1800±n/a nM |
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| Citation |  Gray, NM; Cheng, BK; Mick, SJ; Lair, CM; Contreras, PC Phencyclidine-like effects of tetrahydroisoquinolines and related compounds. J Med Chem32:1242-8 (1989) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Sigma non-opioid intracellular receptor 1 |
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| Name: | Sigma non-opioid intracellular receptor 1 |
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| Synonyms: | Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 25266.54 |
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| Organism: | RAT |
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| Description: | Q9R0C9 |
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| Residue: | 223 |
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| Sequence: | MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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| BDBM50017039 |
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| n/a |
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| Name | BDBM50017039 |
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| Synonyms: | 1-(4-Fluoro-phenyl)-1,2,3,4-tetrahydro-isoquinoline | CHEMBL21277 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H14FN |
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| Mol. Mass. | 227.2768 |
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| SMILES | Fc1ccc(cc1)C1NCCc2ccccc12 |
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| Structure | 
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