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TargetMu-type opioid receptor
LigandBDBM50000784
Substrate/Competitorn/a
Meas. Tech.ChEBML_146255
Ki 702±n/a nM
Citation Cheng, CYWu, SCHsin, LWTam, SW Selective reversible and irreversible ligands for the kappa opioid receptor. J Med Chem35:2243-7 (1992) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50000784
n/a
NameBDBM50000784
Synonyms:2-(3,4-Dichloro-phenyl)-N-methyl-N-(7-pyrrolidin-1-yl-1,4-dioxa-spiro[4.5]dec-8-yl)-acetamide | CHEMBL73226
TypeSmall organic molecule
Emp. Form.C21H28Cl2N2O3
Mol. Mass.427.365
SMILESCN([C@H]1CCC2(C[C@@H]1N1CCCC1)OCCO2)C(=O)Cc1ccc(Cl)c(Cl)c1
Structure
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