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TargetPlatelet-activating factor receptor
LigandBDBM50034231
Substrate/Competitorn/a
Meas. Tech.ChEMBL_162891 (CHEMBL768221)
Temperature310.15±n/a K
IC50>200000±n/a nM
Commentsextracted
Citation Fos, ESuesa, NBorras, LLobato, CBanfi, PGambetta, RAZunino, FMauleón, DCarganico, G Synthesis of alkyl chain-modified ether lipids and evaluation of their in vitro cytotoxicity. J Med Chem38:1216-28 (1995) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Platelet-activating factor receptor
Name:Platelet-activating factor receptor
Synonyms:PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor
Type:Protein
Mol. Mass.:39005.63
Organism:Cavia porcellus
Description:n/a
Residue:342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50034231
n/a
NameBDBM50034231
Synonyms:2-methoxy-3-(7-hexyloctadecyloxy)propyl-2-trimethylammonioethylphosphorate | CHEMBL417824
TypeSmall organic molecule
Emp. Form.C33H70NO6P
Mol. Mass.607.8858
SMILESCCCCCCCCCCCC(CCCCCC)CCCCCCOCC(COP([O-])(=O)OCC[N+](C)(C)C)OC
Structure
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