| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
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| Ligand | BDBM50107597 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_46642 (CHEMBL658898) |
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| Ki | 124±n/a nM |
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| Citation |  López-Rodríguez, ML; Viso, A; Ortega-Gutiérrez, S; Fowler, CJ; Tiger, G; de Lago, E; Fernández-Ruiz, J; Ramos, JA Design, synthesis, and biological evaluation of new inhibitors of the endocannabinoid uptake: comparison with effects on fatty acid amidohydrolase. J Med Chem46:1512-22 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 1 |
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| Name: | Cannabinoid receptor 1 |
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| Synonyms: | Brain-type cannabinoid receptor | CANNABINOID CB1 | CB-R | CB1 | CNR1_RAT | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cnr1 | Skr6 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 52856.55 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | P20272 |
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| Residue: | 473 |
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| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNSPLVPAGDTTNITEFYNKSLSSFKENEENIQCGENFMDMECFMILNPSQQLAI
AVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHV
FHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCL
MWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIVYAYMYILW
KAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPL
LAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTA
QPLDNSMGDSDCLHKHANNTASMHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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| BDBM50107597 |
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| n/a |
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| Name | BDBM50107597 |
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| Synonyms: | (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (1-methyl-1H-pyrrol-2-ylmethyl)-amide | CHEMBL417158 | Icosa-5,8,11,14-tetraenoic acid (1-methyl-1H-pyrrol-2-ylmethyl)-amide |
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| Type | Small organic molecule |
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| Emp. Form. | C26H40N2O |
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| Mol. Mass. | 396.6086 |
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| SMILES | CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)NCc1cccn1C |
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| Structure | 
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