| Reaction Details |
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 | Report a problem with these data |
| Target | Peptide deformylase, mitochondrial |
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| Ligand | BDBM50201872 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_423227 (CHEMBL912248) |
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| IC50 | 450000±n/a nM |
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| Citation |  Boularot, A; Giglione, C; Petit, S; Duroc, Y; Alves de Sousa, R; Larue, V; Cresteil, T; Dardel, F; Artaud, I; Meinnel, T Discovery and refinement of a new structural class of potent peptide deformylase inhibitors. J Med Chem50:10-20 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Peptide deformylase, mitochondrial |
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| Name: | Peptide deformylase, mitochondrial |
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| Synonyms: | DEFM_HUMAN | PDF | PDF1A | Peptide deformylase mitochondrial | Peptide deformylase, mitochondrial | Polypeptide deformylase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 27023.25 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_154318 |
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| Residue: | 243 |
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| Sequence: | MARLWGALSLWPLWAAVPWGGAAAVGVRACSSTAAPDGVEGPALRRSYWRHLRRLVLGPP
EPPFSHVCQVGDPVLRGVAAPVERAQLGGPELQRLTQRLVQVMRRRRCVGLSAPQLGVPR
QVLALELPEALCRECPPRQRALRQMEPFPLRVFVNPSLRVLDSRLVTFPEGCESVAGFLA
CVPRFQAVQISGLDPNGEQVVWQASGWAARIIQHEMDHLQGCLFIDKMDSRTFTNVYWMK
VND
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|
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| BDBM50201872 |
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| n/a |
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| Name | BDBM50201872 |
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| Synonyms: | 2-(5-bromo-2-methyl-1H-indolyl)-N-hydroxyacetamide | CHEMBL219460 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H13BrN2O2 |
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| Mol. Mass. | 297.148 |
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| SMILES | Cc1[nH]c2ccc(Br)cc2c1CC(=O)CNO |
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| Structure | 
|
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