| Reaction Details |
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 | Report a problem with these data |
| Target | P2Y purinoceptor 2 |
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| Ligand | BDBM50378125 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_587771 (CHEMBL1040422) |
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| IC50 | 596000±n/a nM |
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| Citation |  Sauer, R; El-Tayeb, A; Kaulich, M; Müller, CE Synthesis of uracil nucleotide analogs with a modified, acyclic ribose moiety as P2Y(2) receptor antagonists. Bioorg Med Chem17:5071-9 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| P2Y purinoceptor 2 |
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| Name: | P2Y purinoceptor 2 |
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| Synonyms: | ATP receptor | P2RY2_MOUSE | P2U purinoceptor 1 | P2U1 | P2Y purinoceptor 2 | P2Y2 | P2ru1 | P2ry2 | Purinergic receptor | Purinergic receptor P2Y2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42202.78 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_587770 |
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| Residue: | 373 |
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| Sequence: | MAADLEPWNSTINGTWEGDELGYKCRFNEDFKYVLLPVSYGVVCVLGLCLNVVALYIFLC
RLKTWNASTTYMFHLAVSDSLYAASLPLLVYYYARGDHWPFSTVLCKLVRFLFYTNLYCS
ILFLTCISVHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTR
ITCHDTSARELFSHFVAYSSVMLGLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAK
RKSVRTIALVLAVFALCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPLASANSC
LDPVLYFLAGQRLVRFARDAKPPTEPTPSPQARRKLGLHRPNRTVRKDLSVSSDDSRRTE
STPAGSETKDIRL
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| BDBM50378125 |
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| n/a |
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| Name | BDBM50378125 |
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| Synonyms: | CHEMBL572655 |
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| Type | Small organic molecule |
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| Emp. Form. | C8H15N2O12P3 |
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| Mol. Mass. | 424.1322 |
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| SMILES | OP(O)(=O)OP(O)(=O)OP(O)(=O)OCCCCn1ccc(=O)[nH]c1=O |
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| Structure | 
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