| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y-Y2 receptor |
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| Ligand | BDBM50417471 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_687957 (CHEMBL1291629) |
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| Ki | 63.1±n/a nM |
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| Citation |  Lunniss, GE; Barnes, AA; Barton, N; Biagetti, M; Bianchi, F; Blowers, SM; Caberlotto, LL; Emmons, A; Holmes, IP; Montanari, D; Norris, R; Puckey, GV; Walters, DJ; Watson, SP; Willis, J The identification of a series of novel, soluble non-peptidic neuropeptide Y Y2 receptor antagonists. Bioorg Med Chem Lett20:7341-4 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide Y-Y2 receptor |
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| Name: | Neuropeptide Y-Y2 receptor |
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| Synonyms: | n/a |
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| Type: | PROTEIN |
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| Mol. Mass.: | 8731.41 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_687957 |
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| Residue: | 76 |
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| Sequence: | EYSLIEIIPDFEIVACTEKWPGEEKSVYGTVYSLSTLLILYVLPLGIISFSYTRIWSKLK
NHVSPGAASDHYHQRR
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| BDBM50417471 |
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| n/a |
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| Name | BDBM50417471 |
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| Synonyms: | CHEMBL1287953 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H33ClF3N5O |
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| Mol. Mass. | 536.032 |
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| SMILES | CC(C)(C(=O)Nc1ccc(N2CCC3(CCN(CC4CC4)C3)CC2)c(Cl)c1)c1nccc(n1)C(F)(F)F |
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| Structure | 
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