| Reaction Details |
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 | Report a problem with these data |
| Target | Similar to alpha-tubulin isoform 1 |
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| Ligand | BDBM50086304 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1475978 (CHEMBL3428203) |
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| IC50 | 1880±n/a nM |
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| Citation |  Qin, YJ; Li, YJ; Jiang, AQ; Yang, MR; Zhu, QZ; Dong, H; Zhu, HL Design, synthesis and biological evaluation of novel pyrazoline-containing derivatives as potential tubulin assembling inhibitors. Eur J Med Chem94:447-57 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Similar to alpha-tubulin isoform 1 |
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| Name: | Similar to alpha-tubulin isoform 1 |
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| Synonyms: | Similar to alpha-tubulin isoform 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 10383.05 |
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| Organism: | Bos taurus |
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| Description: | ChEMBL_104716 |
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| Residue: | 99 |
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| Sequence: | CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGK
HVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
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| BDBM50086304 |
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| n/a |
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| Name | BDBM50086304 |
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| Synonyms: | CHEMBL3425998 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H26N2O7 |
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| Mol. Mass. | 490.5045 |
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| SMILES | COc1ccc(cc1)C1=NN(C(C1)c1ccc2OCOc2c1)C(=O)c1cc(OC)c(OC)c(OC)c1 |t:9| |
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| Structure | 
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