| Reaction Details |
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 | Report a problem with these data |
| Target | Vasoactive intestinal polypeptide receptor 1 |
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| Ligand | BDBM50435130 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1559802 (CHEMBL3776015) |
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| IC50 | 0.110±n/a nM |
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| Citation |  Waszkielewicz, AM; Gunia-Krzyzak, A; Powroznik, B; Sloczynska, K; Pekala, E; Walczak, M; Bednarski, M; Zeslawska, E; Nitek, W; Marona, H Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents. Bioorg Med Chem24:1793-810 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Vasoactive intestinal polypeptide receptor 1 |
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| Name: | Vasoactive intestinal polypeptide receptor 1 |
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| Synonyms: | VIP 1 | VIPR1 | VIPR1_HUMAN | Vasoactive intestinal polypeptide receptor 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 51557.18 |
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| Organism: | Homo sapiens (Human) |
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| Description: | VIP 1 VIPR1 0::P32241 |
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| Residue: | 457 |
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| Sequence: | MRPPSPLPARWLCVLAGALAWALGPAGGQAARLQEECDYVQMIEVQHKQCLEEAQLENET
IGCSKMWDNLTCWPATPRGQVVVLACPLIFKLFSSIQGRNVSRSCTDEGWTHLEPGPYPI
ACGLDDKAASLDEQQTMFYGSVKTGYTIGYGLSLATLLVATAILSLFRKLHCTRNYIHMH
LFISFILRAAAVFIKDLALFDSGESDQCSEGSVGCKAAMVFFQYCVMANFFWLLVEGLYL
YTLLAVSFFSERKYFWGYILIGWGVPSTFTMVWTIARIHFEDYGCWDTINSSLWWIIKGP
ILTSILVNFILFICIIRILLQKLRPPDIRKSDSSPYSRLARSTLLLIPLFGVHYIMFAFF
PDNFKPEVKMVFELVVGSFQGFVVAILYCFLNGEVQAELRRKWRRWHLQGVLGWNPKYRH
PSGGSNGATCSTQVSMLTRVSPGARRSSSFQAEVSLV
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| BDBM50435130 |
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| n/a |
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| Name | BDBM50435130 |
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| Synonyms: | CHEMBL1893324 |
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| Type | Small organic molecule |
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| Emp. Form. | C147H238N44O42S |
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| Mol. Mass. | 3325.797 |
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| SMILES | n/a |
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| Structure | 
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