Ki Summary BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetFree fatty acid receptor 1
LigandBDBM50180948
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1585169 (CHEMBL3820977)
EC50 7943±n/a nM
Citation Christiansen, EHudson, BDHansen, AHMilligan, GUlven, T Development and Characterization of a Potent Free Fatty Acid Receptor 1 (FFA1) Fluorescent Tracer. J Med Chem59:4849-58 (2016) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Free fatty acid receptor 1
Name:Free fatty acid receptor 1
Synonyms:FFAR1 | FFAR1_HUMAN | G-protein Coupled Receptor 40 | GPR40
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:31473.32
Organism:Homo sapiens (Human)
Description:O14842
Residue:300
Sequence:
MDLPPQLSFGLYVAAFALGFPLNVLAIRGATAHARLRLTPSLVYALNLGCSDLLLTVSLP
LKAVEALASGAWPLPASLCPVFAVAHFFPLYAGGGFLAALSAGRYLGAAFPLGYQAFRRP
CYSWGVCAAIWALVLCHLGLVFGLEAPGGWLDHSNTSLGINTPVNGSPVCLEAWDPASAG
PARFSLSLLLFFLPLAITAFCYVGCLRALARSGLTHRRKLRAAWVAGGALLTLLLCVGPY
NASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGYLGRGPGLKTVCAARTQGGKSQK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50180948
n/a
NameBDBM50180948
Synonyms:CHEBI:30805 | DODECANOATE | Dodecanoic Acid | Dodecanoic Acid Anion | Lauric Acid
TypeSmall organic molecule
Emp. Form.C12H24O2
Mol. Mass.200.3178
SMILESCCCCCCCCCCCC(O)=O
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: