| Reaction Details |
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 | Report a problem with these data |
| Target | Arachidonate 5-lipoxygenase-activating protein |
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| Ligand | BDBM246524 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1664810 (CHEMBL4014606) |
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| Kd | 21000±n/a nM |
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| Citation |  Proschak, E; Heitel, P; Kalinowsky, L; Merk, D Opportunities and Challenges for Fatty Acid Mimetics in Drug Discovery. J Med Chem60:5235-5266 (2017) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Arachidonate 5-lipoxygenase-activating protein |
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| Name: | Arachidonate 5-lipoxygenase-activating protein |
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| Synonyms: | 5-lipoxygenase activating protein | 5-lipoxygenase-activating protein (FLAP) | 5-lipoxygenase/FLAP | AL5AP_HUMAN | ALOX5AP | FLAP | MK-886-binding protein |
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| Type: | Enzyme |
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| Mol. Mass.: | 18159.90 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P20292 |
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| Residue: | 161 |
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| Sequence: | MDQETVGNVVLLAIVTLISVVQNGFFAHKVEHESRTQNGRSFQRTGTLAFERVYTANQNC
VDAYPTFLAVLWSAGLLCSQVPAAFAGLMYLFVRQKYFVGYLGERTQSTPGYIFGKRIIL
FLFLMSVAGIFNYYLIFFFGSDFENYIKTISTTISPLLLIP
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| BDBM246524 |
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| n/a |
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| Name | BDBM246524 |
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| Synonyms: | Psoralidin (5) |
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| Type | Small organic molecule |
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| Emp. Form. | C20H16O5 |
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| Mol. Mass. | 336.338 |
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| SMILES | [#6]\[#6](-[#6])=[#6]\[#6]-c1cc2c3oc4cc(-[#8])ccc4c3c(=O)oc2cc1-[#8] |
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| Structure | 
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