| Reaction Details |
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 | Report a problem with these data |
| Target | Gastrin-releasing peptide |
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| Ligand | BDBM86497 |
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| Substrate/Competitor | n/a |
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| Ki | 110±n/a nM |
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| Comments | PDSP_3737 |
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| Citation |  Mantey, SA; Coy, DH; Entsuah, LK; Jensen, RT Development of bombesin analogs with conformationally restricted amino acid substitutions with enhanced selectivity for the orphan receptor human bombesin receptor subtype 3. J Pharmacol Exp Ther310:1161-70 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Gastrin-releasing peptide |
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| Name: | Gastrin-releasing peptide |
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| Synonyms: | GRP | GRP_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 16223.81 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Gastrin-Releasing peptide 0 HUMAN::P07492 |
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| Residue: | 148 |
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| Sequence: | MRGRELPLVLLALVLCLAPRGRAVPLPAGGGTVLTKMYPRGNHWAVGHLMGKKSTGESSS
VSERGSLKQQLREYIRWEEAARNLLGLIEAKENRNHQPPQPKALGNQQPSWDSEDSSNFK
DVGSKGKVGRLSAPGSQREGRNPQLNQQ
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| BDBM86497 |
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| n/a |
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| Name | BDBM86497 |
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| Synonyms: | CAS_0 | NSC_0 | [D-Tyr6,(S)-Apa11,Phe13,Nle14]Bn(6-14) |
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| Type | Small organic molecule |
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| Emp. Form. | C62H81N16O10 |
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| Mol. Mass. | 1210.4072 |
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| SMILES | CCCC[C@H](NC(=O)[C@H](Cc1ccccc1)N[N+](=N)[C@H](Cc1cnc[nH]1)NC(=O)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](N)Cc1ccc(O)cc1)C(C)C)c1ccccc1)C(N)=O |r| |
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| Structure | 
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