Reaction Details |
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Target | Adenosine receptor A1 |
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Ligand | BDBM86762 |
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Substrate/Competitor | n/a |
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Ki | >10000±n/a nM |
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Comments | PDSP_8527 |
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Citation | Ohshita, K; Ishiyama, H; Oyanagi, K; Nakata, H; Kobayashi, J Synthesis of hybrid molecules of caffeine and eudistomin D and its effects on adenosine receptors. Bioorg Med Chem15:3235-40 (2007) [PubMed] Article |
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More Info.: | Get all data from this article |
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Adenosine receptor A1 |
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Name: | Adenosine receptor A1 |
Synonyms: | A1 adenosine receptor (hA1) | A1AR | AA1R_HUMAN | ADENOSINE A1 | ADORA1 | Adenosine A1 receptor (A1AR) | Adenosine A1-receptor | Adenosine receptor A1 (A1) | Adenosine receptor A1 (hA1) | Adenosine transporter (AdT) |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 36520.92 |
Organism: | Homo sapiens (Human) |
Description: | P30542 |
Residue: | 326 |
Sequence: | MPPSISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKMVVT
PRRAAVAIAGCWILSFVVGLTPMFGWNNLSAVERAWAANGSMGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPSCHKPSILTYIAIFLTHGNSAMNPIVYAFRIQKFRVTFL
KIWNDHFRCQPAPPIDEDLPEERPDD
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BDBM86762 |
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n/a |
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Name | BDBM86762 |
Synonyms: | 2,5,9-trimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione | CAS_44457466 | NSC_44457466 |
Type | Small organic molecule |
Emp. Form. | C12H14N4O2 |
Mol. Mass. | 246.2652 |
SMILES | CN1C2C(N(C)C(=O)N(C)C2=O)c2ncccc12 |
Structure |
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