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TargetMitochondrial peptide methionine sulfoxide reductase
LigandBDBM91498
Substrate/Competitorn/a
Meas. Tech.Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA)
EC50>103909±n/a nM
Citation PubChem, PC Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA) PubChem Bioassay(2012)[AID]
More Info.:Get all data from this article,  Assay Method
 
Mitochondrial peptide methionine sulfoxide reductase
Name:Mitochondrial peptide methionine sulfoxide reductase
Synonyms:MSRA | MSRA protein | MSRA_BOVIN
Type:Enzyme Catalytic Domain
Mol. Mass.:25822.90
Organism:Bos taurus
Description:gi_73586699
Residue:233
Sequence:
MLSATRRALQLFHSLFPIPRMGDSAAKIVSPQEALPGRKEPLVVAAKHHVNGNRTVEPFP
EGTQMAVFGMGCFWGAERKFWTLKGVYSTQVGFAGGYTPNPTYKEVCSGKTGHAEVVRVV
FQPEHISFEELLKVFWENHDPTQGMRQGNDHGSQYRSAIYPTSAEHVGAALKSKEDYQKV
LSEHGFGLITTDIREGQTFYYAEDYHQQYLSKDPDGYCGLGGTGVSCPLGIKK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM91498
n/a
NameBDBM91498
Synonyms:(2S)-2-benzamido-3-methyl-butyric acid (4-keto-5-phenyl-3H-thieno[2,3-d]pyrimidin-2-yl)methyl ester | (2S)-2-benzamido-3-methylbutanoic acid (4-oxo-5-phenyl-3H-thieno[2,3-d]pyrimidin-2-yl)methyl ester | (4-oxidanylidene-5-phenyl-3H-thieno[2,3-d]pyrimidin-2-yl)methyl (2S)-2-benzamido-3-methyl-butanoate | (4-oxo-5-phenyl-3H-thieno[2,3-d]pyrimidin-2-yl)methyl (2S)-2-benzamido-3-methylbutanoate | MLS000339514 | SMR000244129 | cid_2450183
TypeSmall organic molecule
Emp. Form.C25H23N3O4S
Mol. Mass.461.533
SMILESCC(C)[C@H](NC(=O)c1ccccc1)C(=O)OCc1nc2scc(-c3ccccc3)c2c(=O)[nH]1
Structure
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