| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Sigma non-opioid intracellular receptor 1 |
|---|
| Ligand | BDBM93158 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Binding Assay |
|---|
| Ki | 28±0.0 nM |
|---|
| Citation |  Yous, S; Wallez, V; Belloir, M; Caignard, DH; McCurdy, CR; Poupaert, JH Novel 2(3H)-benzothiazolones as highly potent and selective sigma-1 receptor ligands Medicinal Chemistry Research14:158-168 (2005) |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Sigma non-opioid intracellular receptor 1 |
|---|
| Name: | Sigma non-opioid intracellular receptor 1 |
|---|
| Synonyms: | OPRS1 | SGMR1_CAVPO | SIGMAR1 | Sigma 1-type opioid receptor | Sigma non-opioid intracellular receptor 1 | Sigma-1 receptor | Sigma1-receptor | Sigma1R | Sterol isomerase-like protein |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 25307.17 |
|---|
| Organism: | Cavia porcellus (Guinea pig) |
|---|
| Description: | Q60492 |
|---|
| Residue: | 223 |
|---|
| Sequence: | MQWAVGRRWLWVALFLAAVAVLTQIVWLWLGTQNFVFQREEIAQLARQYAGLDHELAFSK
LIVELRRLHPVHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSPRHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLGFALADTVFSTQDFLTLFYTLRVYARALQLELTTYLFGQDP
|
|
|
|---|
| BDBM93158 |
|---|
| n/a |
|---|
| Name | BDBM93158 |
|---|
| Synonyms: | 3-[2-(piperidin-1-yl)ethyl]-6-propyl-2,3-dihydro-1,3-benzoxazol-2-one, 16 |
|---|
| Type | Small molecule |
|---|
| Emp. Form. | C17H24N2O2 |
|---|
| Mol. Mass. | 288.3847 |
|---|
| SMILES | CCCc1ccc2n(CCN3CCCCC3)c(=O)oc2c1 |
|---|
| Structure | 
|
|---|
Search and Browse
