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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Sentrin-specific protease 8 | ||
| Ligand | BDBM71409 | ||
| Substrate/Competitor | n/a | ||
| IC50 | 2040±468 nM | ||
| Citation |  PubChem, PC Dose-response confirmation of uHTS inhibitor hits of Sentrin-Specific Protease 8 using a kinetic assay with Nedd8 Protein Substrate PubChem Bioassay(2012)[AID] | ||
| More Info.: | Get all data from this article | ||
| Sentrin-specific protease 8 | |||
| Name: | Sentrin-specific protease 8 | ||
| Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 24104.52 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | gi_262118306 | ||
| Residue: | 212 | ||
| Sequence: |
| ||
| BDBM71409 | |||
| n/a | |||
| Name | BDBM71409 | ||
| Synonyms: | 2-(2-methoxyphenyl)-4H-isoquinoline-1,3-dione | 2-(2-methoxyphenyl)-4H-isoquinoline-1,3-quinone | MLS001166686 | SMR000592285 | cid_2302144 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C16H13NO3 | ||
| Mol. Mass. | 267.2793 | ||
| SMILES | COc1ccccc1-n1c(O)cc2ccccc2c1=O |(3.08,2.67,;4.41,1.9,;4.41,.36,;3.08,-.41,;3.08,-1.95,;4.41,-2.72,;5.75,-1.95,;5.75,-.41,;7.08,.36,;7.08,1.9,;5.75,2.67,;8.41,2.67,;9.75,1.9,;11.13,2.72,;12.52,1.93,;12.52,.33,;11.13,-.47,;9.75,.36,;8.41,-.41,;8.41,-1.95,)| | ||
| Structure | 
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