| Reaction Details |
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 | Report a problem with these data |
| Target | Protein skinhead-1 |
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| Ligand | BDBM76438 |
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| Substrate/Competitor | n/a |
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| IC50 | 21600±n/a nM |
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| Citation |  PubChem, PC Dose ResponseConfirmation of SKN-1 Inhibitor hits in a fluorescence ratio assay - Set 2 PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article |
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| Protein skinhead-1 |
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| Name: | Protein skinhead-1 |
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| Synonyms: | SKN1_CAEEL | SKiNhead family member (skn-1) | skn-1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 70701.17 |
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| Organism: | Caenorhabditis elegans |
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| Description: | P34707 |
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| Residue: | 623 |
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| Sequence: | MGGSSRRQRSTSATRRDDKRRRRQCFSSVADDEEETTSIYGVSSIFIWILATSSLILVIS
SPSSNTSIQSSSYDRITTKHLLDNISPTFKMYTDSNNRNFDEVNHQHQQEQDFNGQSKYD
YPQFNRPMGLRWRDDQRMMEYFMSNGPVETVPVMPILTEHPPASPFGRGPSTERPTTSSR
YEYSSPSLEDIDLIDVLWRSDIAGEKGTRQVAPADQYECDLQTLTEKSTVAPLTAEENAR
YEDLSKGFYNGFFESFNNNQYQQKHQQQQREQIKTPTLEHPTQKAELEDDLFDEDLAQLF
EDVSREEGQLNQLFDNKQQHPVINNVSLSEGIVYNQANLTEMQEMRDSCNQVSISTIPTT
STAQPETLFNVTDSQTVEQWLPTEVVPNDVFPTSNYAYIGMQNDSLQAVVSNGQIDYDHS
YQSTGQTPLSPLIIGSSGRQQQTQTSPGSVTVTATATQSLFDPYHSQRHSFSDCTTDSSS
TCSRLSSESPRYTSESSTGTHESRFYGKLAPSSGSRYQRSSSPRSSQSSIKIARVVPLAS
GQRKRGRQSKDEQLASDNELPVSAFQISEMSLSELQQVLKNESLSEYQRQLIRKIRRRGK
NKVAARTCRQRRTDRHDKMSHYI
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| BDBM76438 |
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| n/a |
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| Name | BDBM76438 |
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| Synonyms: | 2-(5-bromanylthiophen-2-yl)-6-chloranyl-imidazo[1,2-a]pyridine | 2-(5-bromo-2-thienyl)-6-chloro-imidazo[1,2-a]pyridine | 2-(5-bromo-2-thienyl)-6-chloroimidazo[1,2-a]pyridine | 2-(5-bromo-2-thiophenyl)-6-chloroimidazo[1,2-a]pyridine | 2-(5-bromothiophen-2-yl)-6-chloroimidazo[1,2-a]pyridine | MLS000546882 | SMR000180080 | cid_3850729 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H6BrClN2S |
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| Mol. Mass. | 313.601 |
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| SMILES | Clc1ccc2nc(cn2c1)-c1ccc(Br)s1 |
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| Structure | 
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