| Reaction Details |
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 | Report a problem with these data |
| Target | ADP-ribosylation factor GTPase-activating protein 1 |
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| Ligand | BDBM94700 |
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| Substrate/Competitor | n/a |
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| IC50 | 25560±n/a nM |
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| Citation |  PubChem, PC Fluorescence polarization-based biochemical high throughput dose response screening assay to identify inhibitors of ADP-ribosylation factor GTPase activating protein 1 (ARFGAP1) PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article |
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| ADP-ribosylation factor GTPase-activating protein 1 |
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| Name: | ADP-ribosylation factor GTPase-activating protein 1 |
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| Synonyms: | ARFG1_RAT | Arf1gap | Arfgap1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 45436.38 |
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| Organism: | Rattus norvegicus |
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| Description: | gi_21489979 |
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| Residue: | 415 |
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| Sequence: | MASPRTRKVLKEVRAQDENNVCFECGAFNPQWVSVTYGIWICLECSGRHRGLGVHLSFVR
SVTMDKWKDIELEKMKAGGNAKFREFLEAQDDYEPSWSLQDKYSSRAAALFRDKVATLAE
GKEWSLESSPAQNWTPPQPKTLQFTAHRPAGQPQNVTTSGDKAFEDWLNDDLGSYQGAQE
NRYVGFGNTVPPQKREDDFLNSAMSSLYSGWSSFTTGASKFASAAKEGATKFGSQASQKA
SELGHSLNENVLKPAQEKVKEGRIFDDVSSGVSQLASKVQGVGSKGWRDVTTFFSGKAED
TSDRPLEGHSYQNSSGDNSQNSTIDQSFWETFGSAEPPKAKSPSSDSWTCADASTGRRSS
DSWDIWGSGSASNNKNSNSDGWESWEGASGEGRAKATKKAAPSTAADEGWDNQNW
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| BDBM94700 |
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| n/a |
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| Name | BDBM94700 |
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| Synonyms: | 1,3-bis(o-anisylideneamino)urea | 1,3-bis[(2-methoxyphenyl)methylideneamino]urea | MLS002667206 | SMR001556976 | cid_241318 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H18N4O3 |
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| Mol. Mass. | 326.3498 |
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| SMILES | COc1ccccc1C=NNC(=O)NN=Cc1ccccc1OC |w:14.14,9.10| |
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| Structure | 
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