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Reaction Details
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TargetTrace amine-associated receptor 1
LigandBDBM96724
Substrate/Competitorn/a
IC50 933±n/a nM
Citation PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (hTAAR1): Fluorescence-based cell-based high throughput dose response assay to identify hTAAR1 agonist that also desensitize TAAR1 receptor response. PubChem Bioassay(2013)[AID]
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Trace amine-associated receptor 1
Name:Trace amine-associated receptor 1
Synonyms:TA1 | TAAR1 | TAAR1_HUMAN | TAR1 | TRAR1 | trace amine-associated receptor 1
Type:PROTEIN
Mol. Mass.:39107.47
Organism:Homo sapiens (Human)
Description:ChEMBL_792734
Residue:339
Sequence:
MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNW
LIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISID
RYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRG
GCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNG
ISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFN
PMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
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BDBM96724
n/a
NameBDBM96724
Synonyms:2-(9-phenanthrenyl)guanidine | 2-(9-phenanthryl)guanidine | 2-phenanthren-9-ylguanidine | Guanidine, 1-(9-phenanthryl)- | MLS000757169 | SMR000529028 | cid_344197
TypeSmall organic molecule
Emp. Form.C15H13N3
Mol. Mass.235.2838
SMILES[#7]\[#6](-[#7])=[#7]\c1cc2ccccc2c2ccccc12
Structure
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