Reaction Details |
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Target | Trace amine-associated receptor 1 |
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Ligand | BDBM96761 |
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Substrate/Competitor | n/a |
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IC50 | 1843±n/a nM |
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Citation | PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (hTAAR1): Fluorescence-based cell-based high throughput dose response assay to identify hTAAR1 agonist that also desensitize TAAR1 receptor response. PubChem Bioassay(2013)[AID] |
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More Info.: | Get all data from this article |
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Trace amine-associated receptor 1 |
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Name: | Trace amine-associated receptor 1 |
Synonyms: | TA1 | TAAR1 | TAAR1_HUMAN | TAR1 | TRAR1 | trace amine-associated receptor 1 |
Type: | PROTEIN |
Mol. Mass.: | 39107.47 |
Organism: | Homo sapiens (Human) |
Description: | ChEMBL_792734 |
Residue: | 339 |
Sequence: | MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNW
LIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISID
RYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRG
GCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNG
ISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFN
PMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
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BDBM96761 |
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n/a |
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Name | BDBM96761 |
Synonyms: | 6,8-Dimethyl-3-[(2-m-tolyl-ethylamino)-methyl]-1H-quinolin-2-one | 6,8-dimethyl-3-[[2-(3-methylphenyl)ethylamino]methyl]-1H-quinolin-2-one | 6,8-dimethyl-3-[[2-(m-tolyl)ethylamino]methyl]carbostyril | MLS001204884 | SMR000503420 | cid_3176405 |
Type | Small organic molecule |
Emp. Form. | C21H24N2O |
Mol. Mass. | 320.4281 |
SMILES | Cc1cccc(CCNCc2cc3cc(C)cc(C)c3[nH]c2=O)c1 |
Structure |
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