Ki Summary

Reaction Details

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Target

Guanine nucleotide-binding protein subunit alpha-15

Ligand

BDBM96920

Substrate/Competitor

n/a

IC50

>29908±n/a nM

Citation

PubChem, PC Counterscreen for antagonists of the human trace amine associated receptor 1 (hTAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay(2013)[AID]

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Guanine nucleotide-binding protein subunit alpha-15

Name:

Guanine nucleotide-binding protein subunit alpha-15

Synonyms:

Type:

Protein

Mol. Mass.:

43577.62

Organism:

Homo sapiens (Human)

Description:

P30679

Residue:

374

Sequence:

MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIK
QMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQD
PYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQ
DVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQ
CLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQG
PKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVR
DSVLARYLDEINLL

BDBM96920

n/a

Name

BDBM96920

Synonyms:

4-Amino-isothiazole-3,5-dicarboxylic acid 3-amide 5-{[cyclohexylcarbamoyl-(4-hydroxy-phenyl)-methyl]-o-tolyl-amide} | 4-amino-5-N-[2-(cyclohexylamino)-1-(4-hydroxyphenyl)-2-oxoethyl]-5-N-(2-methylphenyl)-1,2-thiazole-3,5-dicarboxamide | 4-amino-N'-[2-(cyclohexylamino)-1-(4-hydroxyphenyl)-2-keto-ethyl]-N'-(o-tolyl)isothiazole-3,5-dicarboxamide | 4-amino-N5-[2-(cyclohexylamino)-1-(4-hydroxyphenyl)-2-oxoethyl]-N5-(2-methylphenyl)isothiazole-3,5-dicarboxamide | 4-azanyl-N5-[2-(cyclohexylamino)-1-(4-hydroxyphenyl)-2-oxidanylidene-ethyl]-N5-(2-methylphenyl)-1,2-thiazole-3,5-dicarboxamide | MLS001217688 | SMR000599753 | cid_3177673

Type

Small organic molecule

Emp. Form.

C26H29N5O4S

Mol. Mass.

507.605

SMILES

Cc1ccccc1N(C(C(=O)NC1CCCCC1)c1ccc(O)cc1)C(=O)c1snc(C(N)=O)c1N

Structure