| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Guanine nucleotide-binding protein subunit alpha-15 |
|---|
| Ligand | BDBM96930 |
|---|
| Substrate/Competitor | n/a |
|---|
| EC50 | >29881±n/a nM |
|---|
| Citation |  PubChem, PC Counterscreen for antagonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose reponse assay to identify nonselective Ga16 agonists PubChem Bioassay(2013)[AID] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Guanine nucleotide-binding protein subunit alpha-15 |
|---|
| Name: | Guanine nucleotide-binding protein subunit alpha-15 |
|---|
| Synonyms: | G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C] |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 43577.62 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P30679 |
|---|
| Residue: | 374 |
|---|
| Sequence: | MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIK
QMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQD
PYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQ
DVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQ
CLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQG
PKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVR
DSVLARYLDEINLL
|
|
|
|---|
| BDBM96930 |
|---|
| n/a |
|---|
| Name | BDBM96930 |
|---|
| Synonyms: | 2-[(4S,5R)-5-(2-bromophenyl)-4-methyl-4,5,7,8-tetrahydrotriazolo[1,5-d][1,4]oxazepin-3-yl]acetic acid methyl ester | MLS003842904 | SMR002515619 | cid_56588566 | methyl 2-[(4S,5R)-5-(2-bromophenyl)-4-methyl-4,5,7,8-tetrahydro-[1,2,3]triazolo[1,5-d][1,4]oxazepin-3-yl]ethanoate | methyl 2-[(4S,5R)-5-(2-bromophenyl)-4-methyl-4,5,7,8-tetrahydrotriazolo[1,5-d][1,4]oxazepin-3-yl]acetate |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C16H18BrN3O3 |
|---|
| Mol. Mass. | 380.236 |
|---|
| SMILES | COC(=O)Cc1nnn2CCO[C@H]([C@@H](C)c12)c1ccccc1Br |
|---|
| Structure | 
|
|---|
Search and Browse
