| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 3 |
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| Ligand | BDBM62272 |
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| Substrate/Competitor | n/a |
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| IC50 | 143±n/a nM |
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| Citation |  PubChem, PC Fluorescence-based cell-based primary high throughput dose response assay to identify antagonists of the Galanin Receptor 3 (GalR3). PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article |
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| Galanin receptor type 3 |
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| Name: | Galanin receptor type 3 |
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| Synonyms: | GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 39599.97 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Galanin R3 GALR3 HUMAN::O60755 |
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| Residue: | 368 |
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| Sequence: | MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLF
ILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDR
YLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDAR
RRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAV
AALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRA
RFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHG
GEAARGPE
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| BDBM62272 |
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| n/a |
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| Name | BDBM62272 |
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| Synonyms: | MLS-0375912.0001 | N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-methyl-3-pyrazolecarboxamide | N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-methyl-pyrazole-3-carboxamide | N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-methylpyrazole-3-carboxamide | cid_24793159 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H27N5O |
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| Mol. Mass. | 377.4827 |
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| SMILES | Cn1nccc1C(=O)NC1CCCc2c1cnn2-c1ccc(cc1)C(C)(C)C |
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| Structure | 
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