| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 0 group B member 1 |
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| Ligand | BDBM97208 |
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| Substrate/Competitor | n/a |
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| IC50 | >277.93±n/a nM |
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| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): repression of SF-1 (NR5A1) activated StAR promoter by full-length DAX-1 PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article |
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| Nuclear receptor subfamily 0 group B member 1 |
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| Name: | Nuclear receptor subfamily 0 group B member 1 |
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| Synonyms: | AHC | DAX1 | NR0B1 | NR0B1_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 51729.22 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_5016090 |
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| Residue: | 470 |
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| Sequence: | MAGENHQWQGSILYNMLMSAKQTRAAPEAPETRLVDQCWGCSCGDEPGVGREGLLGGRNV
ALLYRCCFCGKDHPRQGSILYSMLTSAKQTYAAPKAPEATLGPCWGCSCGSDPGVGRAGL
PGGRPVALLYRCCFCGEDHPRQGSILYSLLTSSKQTHVAPAAPEARPGGAWWDRSYFAQR
PGGKEALPGGRATALLYRCCFCGEDHPQQGSTLYCVPTSTNQAQAAPEERPRAPWWDTSS
GALRPVALKSPQVVCEAASAGLLKTLRFVKYLPCFQVLPLDQQLVLVRNCWASLLMLELA
QDRLQFETVEVSEPSMLQKILTTRRRETGGNEPLPVPTLQHHLAPPAEARKVPSASQVQA
IKCFLSKCWSLNISTKEYAYLKGTVLFNPDVPGLQCVKYIQGLQWGTQQILSEHTRMTHQ
GPHDRFIELNSTLFLLRFINANVIAELFFRPIIGTVSMDDMMLEMLCTKI
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| BDBM97208 |
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| n/a |
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| Name | BDBM97208 |
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| Synonyms: | 2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2,5-dimethyl-1-(thiophen-2-ylmethyl)pyrrol-3-yl]ethanone | 2-[(5-amino-1,3,4-thiadiazol-2-yl)thio]-1-[2,5-dimethyl-1-(2-thenyl)pyrrol-3-yl]ethanone | 2-[(5-amino-1,3,4-thiadiazol-2-yl)thio]-1-[2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolyl]ethanone | 2-[(5-azanyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2,5-dimethyl-1-(thiophen-2-ylmethyl)pyrrol-3-yl]ethanone | MLS000336319 | SMR000253873 | cid_4880179 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H16N4OS3 |
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| Mol. Mass. | 364.509 |
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| SMILES | Cc1cc(C(=O)CSc2nnc(N)s2)c(C)n1Cc1cccs1 |
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| Structure | 
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