| Reaction Details |
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 | Report a problem with these data |
| Target | Urokinase plasminogen activator surface receptor |
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| Ligand | BDBM98585 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Enzyme Assay |
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| Temperature | 297.15±0 K |
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| Ki | 89±0.0 nM |
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| Citation |  Stuerzebecher, J; Steinmetzer, T; Schweinitz, A Urokinase inhibitors, production and use thereof US Patent US8476306 Publication Date 7/2/2013 |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Urokinase plasminogen activator surface receptor |
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| Name: | Urokinase plasminogen activator surface receptor |
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| Synonyms: | CD87 | Plasminogen activator urokinase | Plaur | U-PAR | UPAR | UPAR_RAT | URKR |
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| Type: | Protein |
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| Mol. Mass.: | 35754.96 |
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| Organism: | Rattus norvegicus |
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| Description: | P49616 |
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| Residue: | 328 |
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| Sequence: | MGLLRRRLLLLVVVVTTCVPASQGLRCIQCESNQDCLVEECALGQDLCRTTVLREWEDAE
ELEVVTRGCAHKEKTNRTMSYRMGSVIVSLTETVCATNLCNRPRPGARGRPFPRGRYLEC
ASCTSLDQSCERGREQSLQCRYPTEHCIEVVTLQSTERSVKDEPYTKGCGSLPGCPGTAG
FHSNQTFHFLKCCNFTQCNGGPVLDLQSLPPNGFQCYSCEGNSTFGCSYEETSLIDCRGP
MNQCLEATGLDVLGNRSYTVRGCATASWCQGSHVADSFQTHVNLSISCCNGSGCNRPTGG
APGPGPAHLILIASLLLTLRLWGIPLWT
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| BDBM98585 |
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| n/a |
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| Name | BDBM98585 |
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| Synonyms: | (2R)-N-[(1S)-2-[(4-carbamimidoylphenyl)methylamino]-1-methyl-2-oxo-ethyl]-2-[(4-cyanophenyl)methylsulfonylamino]-3-hydroxy-propanamide | US8476306, 6.10 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H26N6O5S |
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| Mol. Mass. | 486.544 |
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| SMILES | C[C@H](NC(=O)[C@@H](CO)NS(=O)(=O)Cc1ccc(cc1)C#N)C(=O)NCc1ccc(cc1)C(N)=N |
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| Structure | 
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