| Reaction Details |
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 | Report a problem with these data |
| Target | Urokinase plasminogen activator surface receptor |
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| Ligand | BDBM98604 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Enzyme Assay |
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| Temperature | 297.15±0 K |
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| Ki | 130±0.0 nM |
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| Citation |  Stuerzebecher, J; Steinmetzer, T; Schweinitz, A Urokinase inhibitors, production and use thereof US Patent US8476306 Publication Date 7/2/2013 |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Urokinase plasminogen activator surface receptor |
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| Name: | Urokinase plasminogen activator surface receptor |
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| Synonyms: | CD87 | Plasminogen activator urokinase | Plaur | U-PAR | UPAR | UPAR_RAT | URKR |
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| Type: | Protein |
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| Mol. Mass.: | 35754.96 |
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| Organism: | Rattus norvegicus |
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| Description: | P49616 |
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| Residue: | 328 |
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| Sequence: | MGLLRRRLLLLVVVVTTCVPASQGLRCIQCESNQDCLVEECALGQDLCRTTVLREWEDAE
ELEVVTRGCAHKEKTNRTMSYRMGSVIVSLTETVCATNLCNRPRPGARGRPFPRGRYLEC
ASCTSLDQSCERGREQSLQCRYPTEHCIEVVTLQSTERSVKDEPYTKGCGSLPGCPGTAG
FHSNQTFHFLKCCNFTQCNGGPVLDLQSLPPNGFQCYSCEGNSTFGCSYEETSLIDCRGP
MNQCLEATGLDVLGNRSYTVRGCATASWCQGSHVADSFQTHVNLSISCCNGSGCNRPTGG
APGPGPAHLILIASLLLTLRLWGIPLWT
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| BDBM98604 |
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| n/a |
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| Name | BDBM98604 |
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| Synonyms: | 2-[4-[[(1R)-2-[[2-[4-[(3-amino-4-methoxy-benzoyl)amino]anilino]-2-oxo-ethyl]amino]-1-(hydroxymethyl)-2-oxo-ethyl]sulfamoylmethyl]phenyl]acetic acid | US8476306, 13 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H27N5O7S |
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| Mol. Mass. | 505.544 |
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| SMILES | NC(=N)c1ccc(CNC(=O)CNC(=O)[C@H](CO)NS(=O)(=O)Cc2ccc(CC(O)=O)cc2)cc1 |
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| Structure | 
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