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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Carboxypeptidase B2 | ||
| Ligand | BDBM109244 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Enzyme Inhibition Assay | ||
| IC50 | 19±n/a nM | ||
| Citation |  Nagata, T; Inoue, M; Ashida, Y; Noguchi, K; Ono, M Cycloalkyl-substituted imidazole derivative US Patent US8609710 Publication Date 12/17/2013 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Carboxypeptidase B2 | |||
| Name: | Carboxypeptidase B2 | ||
| Synonyms: | CBPB2_HUMAN | CPB2 | CPU | Carboxypeptidase B2 | Carboxypeptidase B2 isoform A | Carboxypeptidase U | Plasma carboxypeptidase B | TAFI | Thrombin-activable fibrinolysis inhibitor | pCPB | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 48432.74 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | Q96IY4 | ||
| Residue: | 423 | ||
| Sequence: |
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| BDBM109244 | |||
| n/a | |||
| Name | BDBM109244 | ||
| Synonyms: | US8609710, 8 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C16H27N3O3 | ||
| Mol. Mass. | 309.4039 | ||
| SMILES | CC1(O)CCC(CC1)n1cnc(CC(CCCN)C(O)=O)c1 |(-4.54,4.74,;-3.45,3.65,;-3.05,5.14,;-1.97,3.25,;-1.57,1.76,;-2.66,.68,;-4.14,1.07,;-4.54,2.56,;-2.26,-.81,;-3.16,-2.06,;-2.26,-3.3,;-.79,-2.83,;.54,-3.6,;1.87,-2.83,;1.87,-1.29,;3.21,-.52,;3.21,1.02,;4.54,1.79,;3.21,-3.6,;3.21,-5.14,;4.54,-2.83,;-.79,-1.29,)| | ||
| Structure | 
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