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TargetNuclear hormone receptor family member daf-12
LigandBDBM114772
Substrate/Competitorn/a
Meas. Tech.Luminescence-based cell-based high throughput dose response assay to identify agonists of the DAF-12 from the parasite H. contortus (hcDAF-12)
EC50 67541±n/a nM
Citation PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify agonists of the DAF-12 from the parasite H. contortus (hcDAF-12) PubChem Bioassay(2013)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Nuclear hormone receptor family member daf-12
Name:Nuclear hormone receptor family member daf-12
Synonyms:DAF12_CAEEL | Protein DAF-12, isoform a | XL285 | daf-12 | daf-20 | mig-7
Type:Enzyme Catalytic Domain
Mol. Mass.:84211.49
Organism:Caenorhabditis elegans
Description:gi_71987181
Residue:753
Sequence:
MGTNGGVIAEQSMEIETNENPDKVEEPVVRRKRVTRRRHRRIHSKNNCLTPPNSDDDPQM
STPDDPVIHSPPSIGAAPGMNGYHGSGVKLEESSGACGSPDDGLLDSSEESRRRQKTCRV
CGDHATGYNFNVITCESCKAFFRRNALRPKEFKCPYSEDCEINSVSRRFCQKCRLRKCFT
VGMKKEWILNEEQLRRRKNSRLNNTGTCNKRSQPGNQQSPQGPNQQPHLSPHHPGVAIYP
PQPQRPLTINPMDNQMMHHMQANRPNAMPQLISPPGAQPYPLTSPVGSSASDSPPNRSLT
MMHNGEKSPDGYDPNIMAHRAPPPSFNNRPKMDSGQVVLSTEEYKQLLSRIPGAQVPGLM
NEEEPINKRAAYNCNGHPMPAETTPPYSAPMSDMSLSRHNSTSSGTEKNHMTHSTVSAIP
GNSAQNHFDIASFGMGIVTATGGGDAAEEMYKRMNMFYENCIQSALDSPENQEPKPQEAM
IPKEEYMTPTHGFQYQSDPYQVPPAERNINYQLNAAELKALDAVREAFYGMDDPMEQGRQ
MQSFLKANKTPADIMNIMDVTMRRFVKVAKGVPAFREVSQEGKFSLLKGGMIEMLTVRGV
TRYDASTNSFKTPTIKGQNVSVNVDDMFAKLNANAQAQKAKCLEFFGFFDEEIKKNELAV
YLVMLAVLFSVRSDPPMNENDVRIVTERHNHFMSLLNRYLESLFGEQARRIFERIPKALG
LLNEIARNAGMLFMGTVRSGEAEELPGEFFKIK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM114772
n/a
NameBDBM114772
Synonyms:(2Z)-2-(phenylhydrazinylidene)-1-benzothiophen-3-one | (2Z)-2-(phenylhydrazono)benzothiophen-3-one | 2-(Phenyl-hydrazono)-benzo[b]thiophen-3-one | MLS000777106 | SMR000413502 | cid_5419037
TypeSmall organic molecule
Emp. Form.C14H10N2OS
Mol. Mass.254.307
SMILESOc1c(N=Nc2ccccc2)sc2ccccc12 |w:3.2|
Structure
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