| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 4 |
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| Ligand | BDBM123486 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radio Ligand Binding Assay |
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| pH | 8±n/a |
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| IC50 | 38±n/a nM |
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| Citation |  Miltz, W; Oberhauser, B; Vaupel, A; Velcicky, J; Weigand, K; Leleti, RR; Liu, Y; Du, Z Pyrazolo pyrimidine derivatives US Patent US8748435 Publication Date 6/10/2014 |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| G-protein coupled receptor 4 |
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| Name: | G-protein coupled receptor 4 |
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| Synonyms: | G-protein coupled receptor 4 | G-protein coupled receptor 4 (GPR4) | GPR4 | GPR4_HUMAN |
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| Type: | Enzyme |
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| Mol. Mass.: | 40994.40 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P46093 |
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| Residue: | 362 |
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| Sequence: | MGNHTWEGCHVDSRVDHLFPPSLYIFVIGVGLPTNCLALWAAYRQVQQRNELGVYLMNLS
IADLLYICTLPLWVDYFLHHDNWIHGPGSCKLFGFIFYTNIYISIAFLCCISVDRYLAVA
HPLRFARLRRVKTAVAVSSVVWATELGANSAPLFHDELFRDRYNHTFCFEKFPMEGWVAW
MNLYRVFVGFLFPWALMLLSYRGILRAVRGSVSTERQEKAKIKRLALSLIAIVLVCFAPY
HVLLLSRSAIYLGRPWDCGFEERVFSAYHSSLAFTSLNCVADPILYCLVNEGARSDVAKA
LHNLLRFLASDKPQEMANASLTLETPLTSKRNSTAKAMTGSWAATPPSQGDQVQLKMLPP
AQ
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| BDBM123486 |
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| n/a |
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| Name | BDBM123486 |
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| Synonyms: | US8748435, 11 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H34N6O |
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| Mol. Mass. | 446.5878 |
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| SMILES | CCc1nn2c(C)cc(C)nc2c1Cc1ccc(\C=C\CN2CCN(CC2)C(=O)CN)cc1 |
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| Structure | 
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