Reaction Details |
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Target | Transthyretin |
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Ligand | BDBM128232 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Luminescence-based cell-based high throughput dose response assay to identify activators of Transthyretin (TTR) transcription |
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EC50 | >167158±n/a nM |
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Citation | PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify activators of Transthyretin (TTR) transcription PubChem Bioassay(2014)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Transthyretin |
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Name: | Transthyretin |
Synonyms: | ATTR | PALB | Prealbumin | TBPA | TTHY_HUMAN | TTR | Transthyretin (TTR) |
Type: | Enzyme |
Mol. Mass.: | 15884.31 |
Organism: | Homo sapiens (Human) |
Description: | P02766 |
Residue: | 147 |
Sequence: | MASHRLLLLCLAGLVFVSEAGPTGTGESKCPLMVKVLDAVRGSPAINVAVHVFRKAADDT
WEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDS
GPRRYTIAALLSPYSYSTTAVVTNPKE
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BDBM128232 |
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n/a |
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Name | BDBM128232 |
Synonyms: | 3-(3,4-Dimethoxy-phenyl)-5-thiophen-2-yl-[1,2,4]oxadiazole | 3-(3,4-dimethoxyphenyl)-5-(2-thienyl)-1,2,4-oxadiazole | 3-(3,4-dimethoxyphenyl)-5-thiophen-2-yl-1,2,4-oxadiazole | MLS000333489 | SMR000437691 | cid_1221653 |
Type | Small organic molecule |
Emp. Form. | C14H12N2O3S |
Mol. Mass. | 288.322 |
SMILES | COc1ccc(cc1OC)-c1noc(n1)-c1cccs1 |
Structure |
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