| Reaction Details |
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 | Report a problem with these data |
| Target | Transthyretin |
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| Ligand | BDBM128234 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Luminescence-based cell-based high throughput dose response assay to identify activators of Transthyretin (TTR) transcription |
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| EC50 | >167158±n/a nM |
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| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify activators of Transthyretin (TTR) transcription PubChem Bioassay(2014)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Transthyretin |
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| Name: | Transthyretin |
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| Synonyms: | ATTR | PALB | Prealbumin | TBPA | TTHY_HUMAN | TTR | Transthyretin (TTR) |
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| Type: | Enzyme |
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| Mol. Mass.: | 15884.31 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P02766 |
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| Residue: | 147 |
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| Sequence: | MASHRLLLLCLAGLVFVSEAGPTGTGESKCPLMVKVLDAVRGSPAINVAVHVFRKAADDT
WEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDS
GPRRYTIAALLSPYSYSTTAVVTNPKE
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| BDBM128234 |
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| n/a |
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| Name | BDBM128234 |
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| Synonyms: | (5-bromopyrimidin-2-yl)-[(E)-1-(3-nitrophenyl)ethylideneamino]amine | 5-bromanyl-N-[(E)-1-(3-nitrophenyl)ethylideneamino]pyrimidin-2-amine | 5-bromo-N-[(E)-1-(3-nitrophenyl)ethylideneamino]-2-pyrimidinamine | 5-bromo-N-[(E)-1-(3-nitrophenyl)ethylideneamino]pyrimidin-2-amine | MLS001211234 | N-(5-Bromo-pyrimidin-2-yl)-N'-[1-(3-nitro-phenyl)-ethylidene]-hydrazine | SMR000513413 | cid_5338790 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H10BrN5O2 |
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| Mol. Mass. | 336.144 |
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| SMILES | C\C(=N/Nc1ncc(Br)cn1)c1cccc(c1)[N+]([O-])=O |
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| Structure | 
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