| Reaction Details |
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 | Report a problem with these data |
| Target | Fatty acid-binding protein 5 |
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| Ligand | BDBM212450 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Time Resolved-Fluorescence Energy Transfer (TR-FRET) Assay |
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| pH | 7.5±n/a |
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| Temperature | 298.15±n/a K |
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| IC50 | >50000±n/a nM |
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| Comments | extracted |
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| Citation |  Buettelmann, B; Ceccarelli, SM; Conte, A; Kuehne, H; Kuhn, B; Neidhart, W; Obst Sander, U; Richter, H Urea derivatives and their use as fatty-acid binding protein (FABP) inhibitors US Patent US9278918 Publication Date 3/8/2016 |
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| More Info.: | Get all data from this article, Assay Method |
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| Fatty acid-binding protein 5 |
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| Name: | Fatty acid-binding protein 5 |
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| Synonyms: | FABP5 | FABP5_HUMAN | Fatty acid binding protein epidermal | Fatty acid-binding protein 5 (FABP5) |
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| Type: | Enzyme |
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| Mol. Mass.: | 15164.79 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q01469 |
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| Residue: | 135 |
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| Sequence: | MATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTL
KTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVEC
VMNNVTCTRIYEKVE
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| BDBM212450 |
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| n/a |
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| Name | BDBM212450 |
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| Synonyms: | US9278918, 40 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H14ClFN2O3 |
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| Mol. Mass. | 348.756 |
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| SMILES | OC(=O)C1(CC1)NC(=O)Nc1cc(Cl)ccc1-c1ccc(F)cc1 |
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| Structure | 
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