| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 4 group A member 1 |
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| Ligand | BDBM40631 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters |
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| IC50 | 16524±2100 nM |
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| Citation |  PubChem, PC High Throughput Fluorescence Polarization Screen for Bcl-B Phenotype Converters PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Nuclear receptor subfamily 4 group A member 1 |
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| Name: | Nuclear receptor subfamily 4 group A member 1 |
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| Synonyms: | GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 64467.13 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_27894344 |
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| Residue: | 598 |
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| Sequence: | MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
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| BDBM40631 |
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| n/a |
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| Name | BDBM40631 |
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| Synonyms: | 2-(5,6-dihydro-4H-cyclopent[d]isoxazole-3-carbonylamino)benzoic acid methyl ester | 2-[[5,6-dihydro-4H-cyclopenta[d]isoxazol-3-yl(oxo)methyl]amino]benzoic acid methyl ester | MLS000087339 | SMR000023562 | cid_3240336 | methyl 2-(5,6-dihydro-4H-cyclopenta[d][1,2]oxazol-3-ylcarbonylamino)benzoate | methyl 2-(5,6-dihydro-4H-cyclopenta[d][1,2]oxazole-3-carbonylamino)benzoate | methyl 2-[(5,6-dihydro-4H-cyclopenta[d]isoxazol-3-ylcarbonyl)amino]benzoate |
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| Type | Small organic molecule |
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| Emp. Form. | C15H14N2O4 |
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| Mol. Mass. | 286.2827 |
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| SMILES | COC(=O)c1ccccc1NC(=O)c1noc2CCCc12 |
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| Structure | 
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